The organocatalytic two-step synthesis of diversely functionalized tricyclic tetrazoles.

نویسندگان

  • Xiong Huang
  • Ping Li
  • Xin-Sheng Li
  • Dong-Cheng Xu
  • Jian-Wu Xie
چکیده

The diversely functionalized tricyclic tetrazoles were synthesised from readily available substrates via intramolecular 1,3-dipolar cycloaddition as the key step in good yields (53-78% yield for two steps) with high enantioselectivities (81-99% ee).

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 8 20  شماره 

صفحات  -

تاریخ انتشار 2010